Staff Members - Benha University
Benzotriazole-Assisted Thioacylation
J. Org. Chem. • 2005
Publication Information
Authors
Alan R. Katritzky,*,§ Rachel M. Witek,§ Valerie Rodriguez-Garcia,§ Prabhu P. Mohapatra,§
James W. Rogers,§ Janet Cusido,§ Ashraf A. A. Abdel-Fattah,§ and Peter J. Steel|
Keywords
Not Available
Journal
J. Org. Chem.
Publisher
American Chemical Society
Volume
70
Issue
Not Available
Pages
7866-7881
publication.type
International
Paper Link
Not Available
Supplementary Materials
Not Available
Abstract
Benzotriazole reagents for thioacylation (RCSBt), thiocarbamoylation (RR¢NCSBt), aryl/alkoxythioacylation
(ROCSBt), and aryl/alkylthiothioacylation (RSCSBt) are synthesized, and their utility
is assessed by syntheses of representative heteroaryl thioureas 3a-g, thioamides 15a-s, thionoesters
16a-h, thiocarbamates 17a-e, dithiocarbamates 18a-d, thiocarbonates 19a-c, and
dithiocarbonates 20a-c.
(ROCSBt), and aryl/alkylthiothioacylation (RSCSBt) are synthesized, and their utility
is assessed by syntheses of representative heteroaryl thioureas 3a-g, thioamides 15a-s, thionoesters
16a-h, thiocarbamates 17a-e, dithiocarbamates 18a-d, thiocarbonates 19a-c, and
dithiocarbonates 20a-c.