| publication name | Benzotriazole-Assisted Thioacylation |
|---|---|
| Authors | Alan R. Katritzky,*,§ Rachel M. Witek,§ Valerie Rodriguez-Garcia,§ Prabhu P. Mohapatra,§ James W. Rogers,§ Janet Cusido,§ Ashraf A. A. Abdel-Fattah,§ and Peter J. Steel| |
| year | 2005 |
| keywords | |
| journal | J. Org. Chem. |
| volume | 70 |
| issue | Not Available |
| pages | 7866-7881 |
| publisher | American Chemical Society |
| Local/International | International |
| Paper Link | Not Available |
| Full paper | download |
| Supplementary materials | Not Available |
Abstract
Benzotriazole reagents for thioacylation (RCSBt), thiocarbamoylation (RR¢NCSBt), aryl/alkoxythioacylation (ROCSBt), and aryl/alkylthiothioacylation (RSCSBt) are synthesized, and their utility is assessed by syntheses of representative heteroaryl thioureas 3a-g, thioamides 15a-s, thionoesters 16a-h, thiocarbamates 17a-e, dithiocarbamates 18a-d, thiocarbonates 19a-c, and dithiocarbonates 20a-c.